AKR1C3-IN-6

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AKR1C3-IN-6

本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

CAS NO:

2137881-54-8

AKR1C3-IN-6 (Compound 1) 是一种有效的、选择性的AKR1C3抑制剂，对 AKR1C3 和AKR1C2的IC₅₀分别为 0.31 μM 和 73.23 μM。AKR1C3-IN-6 具有抗肿瘤活性。

生物活性	AKR1C3-IN-6 (Compound 1) is a potent, selectiveAKR1C3inhibitor withIC₅₀values of 0.31 μM and 73.23 μM against AKR1C3 andAKR1C2, respectively. AKR1C3-IN-6 shows antitumor activity^[1].
IC₅₀& Target	IC₅₀: 0.31 μM (AKR1C3), 73.23 μM (AKR1C2)^[1]
体外研究 (In Vitro)	AKR1C3-IN-6 (Compound 1) shows antiproliferative activity with an IC₅₀of 81.40 ± 2.29 μM against prostate cancer cell line 22rv1^[1].
分子量	392.33
Formula	C₁₈H₁₅F₃N₄O₃
CAS 号	2137881-54-8
运输条件	Room temperature in continental US; may vary elsewhere.
储存方式	Please store the product under the recommended conditions in the Certificate of Analysis.