CS-2100 (Compound 10b) 是一种有效的、选择性的、口服活性的 S1P3-sparingS1P1激动剂，对人 S1P1的EC50值为 4.0 nM。CS-2100在大鼠体内具有免疫抑制效果，对 HvGR 的ID50值为 0.407 mg/kg。
| 生物活性 | CS-2100 (Compound 10b) is a potent, selective, orally active and S1P3-sparingS1P1agonist with anEC50of 4.0 nM for human S1P1. CS-2100 shows in vivo immunosuppressive efficacy in rats with anID50(infective dose) of 0.407 mg/kg for HvGR[1]. |
| IC50& Target | EC50: 4.0 nM (human S1P1)[1] |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
