CB2 receptor agonist 3 是一种稳健和选择性的CB2大麻素激动剂，对 CB2 和 CB1 的Ki分别为 7.6 和 900 nM。CB2 receptor agonist 3 显著增加 HL-60 细胞 P-ERK1/2 的表达。
| 生物活性 | CB2receptor agonist 3 is a robust and selectiveCB2cannabinoid agonist withKis of 7.6 and 900 nM forCB2andCB1, respectively.CB2receptor agonist 3 significantly increases P-ERK 1/2 expression in HL-60 cells[1]. |
体外研究
(In Vitro) | CB2 receptor agonist 3 (Compound 2a) is also shown to be agonist in an in vitro model based on human promyelocytic leukemia HL-60 cells[1].
|
| 分子量 | |
| 性状 | |
| Formula | |
| CAS 号 | |
| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | | Powder | -20°C | 3 years | | 4°C | 2 years | | In solvent | -80°C | 6 months | | -20°C | 1 month |
|
