HS 024 是一种选择性 MC4 受体拮抗剂，对 MC4、MC5、MC3 和 MC1 的 Kis 分别为 0.29、3.29、5.45 和 18.6 nM。
| Cas No. | 212370-59-7 |
| Canonical SMILES | CCCC[C@@](/N=C(O)/[C@](/N=C(O)/C)([H])CS)([H])/C(O)=N/[C@@](/C(O)=N/[C@@](/C(O)=N/[C@](/C(O)=N/[C@@](/C(O)=N/[C@@](/C(O)=N/C/C(O)=N/[C@@](C(O)=N)([H])CS)([H])CC1=CNC2=CC=CC=C12)([H])CCCNC(N)=N)([H])CC3=CC4=CC=CC=C4C=C3)([H])CC5=CN=CN5)([H])CCCNC(N)=N |
| 分子式 | C58H79N19O10S2 |
| 分子量 | 1266.5 |
| 溶解度 | Soluble to 0.50 mg/ml in Water |
| 储存条件 | Desiccate at -20°C |
| General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
| Shipping Condition | Evaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request |
