PSB36 是一种有效和选择性的腺苷 A1受体 (adenosine A1receptor) 拮抗剂，对rA1,hA2B,rA2A,hA3和rA3的Ki值分别为 0.12 nM, 187 nM, 552 nM, 2300 nM 和 6500 nM。PSB36 可用于痛觉过敏的研究。
| 生物活性 | PSB36 is a potent and selective antagonist ofadenosine A1receptor, withKis 0.12 nM, 187 nM, 552 nM, 2300 nM, and 6500 nM forrA1,hA2B,rA2A,hA3andrA3receptorsrespectively. PSB36 can be used for the research of hyperalgesia[1][2]. |
| IC50& Target[1] | rA1 0.12 nM (Ki) | hA2B 187 nM (Ki) | rA2A 552 nM (Ki) | hA3 2300 nM (Ki) | rA3 6500 nM (Ki) |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
