hMC1R agonist 1 是一种有效的选择性hMC1R激动剂(EC50=3 nM)，hMC1R agonist 1 对hMC1R的选择性是hMC3R(b>EC50=902 nM),hMC4R(b>EC50=915 nM), 和hMC5R(b>EC50=>1000 nM) 的 300 倍。hMC1R agonist 1 有治疗和预防黑皮质素家族疾病的潜能。
| 生物活性 | (EC50=3 nM). hMC1R agonist 1 shows at least 300-fold selectivity forhMC1RoverhMC3R(b>EC50=902 nM),hMC4R(b>EC50=915 nM), andhMC5R(b>EC50=>1000 nM). hMC1R agonist 1 has the potential for the therapeutic intervention of melanocortin family[1]. |
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| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
