ZJ43 是一种有效的NAAG肽酶抑制剂，其IC50为 2.4 nM，Ki为 0.8 nM。ZJ43 能充分激活 II 组 mGluR，降低 PCP 的部分行为效应。ZJ43 在神经病变、炎症和疼痛模型中具有镇痛作用。
| 生物活性 | ZJ43 is a potentNAAG peptidaseinhibitor, with anIC50of 2.4 nM and a Kiof 0.8 nM. ZJ43 sufficiently activates group IImGluRand reduces some of the behavioral effects of PCP. ZJ43 shows an analgesic effect in neuropathic and inflammatory and pain models[1]. |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
