PHCCC(4Me) (THCCC) 是一种 PHCCC 类似物，是一种双重mGluR2(IC50为 1.5 μM) 负变构调节剂和mGluR3(EC50为 8.9 μM) 正变构调节剂。
| 生物活性 | PHCCC(4Me) (THCCC), a PHCCC analog, is a dualmGluR2(IC50of 1.5 μM) negative allosteric modulator andmGluR3(EC50of 8.9 μM) positive allosteric modulator[1]. |
体外研究
(In Vitro) | PHCCC(4Me) (THCCC; Compound 3) shows micromolar affinity
for mGluR2, with a Kivalue of 0.6 μM[1].
|
| 分子量 | |
| Formula | |
| CAS 号 | |
| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
