mGluR2 modulator 3

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mGluR2 modulator 3

本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

CAS NO:

1004614-58-7

mGluR2 modulator 3 (compound 1) 是一种有效的mGluR2正向变构调节剂，EC₅₀为 0.87 μM。mGluR2 modulator 3 在精神疾病模型中具有体内活性，如在小鼠中甲基苯丙胺诱导的多动症和 Mescaline 诱导的抓挠症。

生物活性

mGluR2 modulator3 (compound 1) is a potentmGluR2positive allosteric modulator with anEC₅₀value of 0.87 μM.mGluR2 modulator3 has activity in psychosis disease models such as methamphetamine-induced hyperactivity and mescaline-induced scratching in mice^[1].

IC₅₀& Target^[1]

mGluR2

0.87 μM (EC₅₀)

分子量

335.44

Formula

C₂₁H₂₅N₃O

CAS 号

1004614-58-7

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.