BIBP3226 是一种有效选择性的神经肽 Y Y1(NPY Y1)和神经肽 FF(NPFF)受体拮抗剂，对 rNPY Y1，hNPFF2，rNPFF 的Ki分别为 1.1、79、108 nM。BIBP3226 具有焦虑样作用。
| 生物活性 | BIBP3226 is a potent and selective neuropeptide Y Y1(NPY Y1)and neuropeptide FF(NPFF) receptorantagonist, withKis of 1.1, 79, and 108 nM for rNPY Y1, hNPFF2, and rNPFF, respectively. BIBP3226 displays anxiogenic-like effect[1][2]. |
体内研究
(In Vivo) | BIBP3226 (0.5, 5 μg; i.c.v.; male Wistar rats) induces an anxiogenic-like effect at the higher dose[1].
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
