(S)-Sitagliptin phosphate

立即咨询

本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

CAS NO:

823817-58-9

(S)-MK-0431 phosphate

(S)-Sitagliptin phosphate 是 Sitagliptin phosphate 的低活性 S 型异构体。Sitagliptin phosphate (MK-0431 phosphate) 是一种有效的 DPP4 抑制剂，在 Caco-2 细胞中， IC₅₀值为 19 nM。

生物活性

(S)-Sitagliptin phosphate is the less active S-enantiomer of Sitagliptin phosphate. Sitagliptin phosphate (MK-0431 phosphate) is a potent inhibitor of DPP4 with an IC₅₀of 19 nM in Caco-2 cell extracts^[1].

IC₅₀& Target

DPP-4

分子量

505.31

Formula

C₁₆H₁₈F₆N₅O₅P

CAS 号

823817-58-9

中文名称

西格列汀/西他列汀EP杂质A Phosphate

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.