FASN-IN-4 是高效的脂肪酸合酶FASN抑制剂，IC50值为 10 nM (WO2012064642A1, compound 29)。FASN-IN-4 还抑制SARS-CoV-2，EC50为 18.6 nM。
| 生物活性 | FASN-IN-4 is a potent inhibitor offatty acid synthase(FASN) with anIC50of 10 nM (WO2012064642A1, compound 29)[1]. FASN-IN-4 also inhibitsSARS-CoV-2with anEC50of 18.6 nM[2]. |
| IC50& Target | IC50: 10 nM (FASN)[1]
EC50: 18.6 nM (SARS-CoV-2)[2] |
体外研究
(In Vitro) | The FASN inhibitor, FASN-IN-4 inhibits SARS-CoV-2 replication, and has the potential for COVID-19 research[2].
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | | Powder | -20°C | 3 years | | 4°C | 2 years | | In solvent | -80°C | 6 months | | -20°C | 1 month |
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