IDO1/2-IN-1 是第一个有效的IDO1/IDO2双重抑制剂，对 IDO1 和 IDO2 的IC50分别为 28 nM 和 144 nM。IDO1/2-IN-1 具有抗肿瘤活性。具有口服活性。
| 生物活性 | IDO1/2-IN-1 (compound 4t) is the first potentIDO1/IDO2dual inhibitor withIC50s of 28 nM and 144 nM forIDO1andIDO2, respectively. IDO1/2-IN-1 exhibits antitumor activies. Orally active[1]. |
| IC50& Target[1] | IDO1 28 nM (IC50) | IDO2 144 nM (IC50) |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
