MMP-2/9-IN-1 (Compound 4a) 是一种有效的MMP-2和MMP-9双重抑制剂,其IC50值分别为 56 nM 和 38 nM。MMP-2/9-IN-1 抑制肿瘤生长,强烈诱导癌细胞凋亡 (apoptosis),抑制细胞迁移,抑制细胞周期进程导致 DNA 片段化
生物活性 | MMP-2/9-IN-1 (Compound 4a) is a potent dualMMP-2andMMP-9inhibitor withIC50values of 56 nM and 38 nM, respectively. MMP-2/9-IN-1 inhibits tumor growth, strongly inducescancercellapoptosis, inhibits cell migration, and suppresses cell cycle progression leading to DNA fragmentation[1]. |
IC50& Target | MMP-2 56 nM (IC50) | MMP-9 38 nM (IC50) |
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运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |