LSD1-IN-17

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LSD1-IN-17

本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

LSD1-IN-17 (compound 5b) 是一种有效的LSD1抑制剂。LSD1-IN-17 对LSD1-CoREST、MAO-A和MAO-B具有抑制作用，IC₅₀值分别为 0.005、0.028 和 0.820 μM。LSD1-IN-17 在前列腺癌 LNCaP 细胞中显示细胞生长阻滞，IC₅₀为 17.2 μM。

生物活性

LSD1-IN-17 (compound 5b) is a potentLSD1inhibitor. LSD1-IN-17 can inhibitLSD1-CoREST,MAO-AandMAO-B, withIC₅₀values of 0.005, 0.028, and 0.820 μM, respectively. LSD1-IN-17 displays cell growth arrest in prostatecancerLNCaP cells, with anIC₅₀of 17.2 μM^[1].

IC₅₀& Target

MAO-A

0.028 ± 0. μM (IC₅₀)

MAO-B

0.820 ± 0. μM (IC₅₀)

分子量

334.43

Formula

C₂₀H₁₈N₂OS

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.