OMDM-6 是VR1 (TRPV1)受体 (EC50=75 nM) 和大麻素 1 型受体(CB1)(Ki=3.2 μM) 的混合激动剂。OMDM-6 抑制 anandamide 细胞摄取(ACU)，Ki为 7.0 μM。
| 生物活性 | OMDM-6 is a hybrid agonist ofvanilloid receptor type 1 (VR1, TRPV1)(EC50=75 nM) andcannabinoid receptortype 1 (CB1)(Ki=3.2 μM). OMDM-6 inhibitsanandamide cellular uptake (ACU)with aKiof 7.0 μM[1]. |
| IC50& Target | EC50: 75 nM (vanilloid receptor type 1), Ki: 3.2 μM (cannabinoid receptor type 1), Ki: 7.0 μM (anandamide cellular uptake)[1] |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
