Tiagabine (NO050328) 是一种有效、选择性的GABA reuptake抑制剂，为抗惊厥剂；在突触体、神经元和神经胶质中，能够抑制 [3H]GABA 的重摄取，IC50值分别为 67，446 和 182 nM。
| 生物活性 | Tiagabine (NO050328) is a potent and selectiveGABA reuptakeinhibitor, used as an anticonvulsant agent, withIC50s of 67, 446 and 182 nM for [3H]GABA uptake in Synaptosomes, Neurons and Glia, respectively[1]. |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
