Raloxifene 6-Monomethyl Ether 是一种 Raloxifene 衍生物，其抑制雌激素受体 α (estrogen receptor α)。Raloxifene 4-Monomethyl Ether 抑制 MCF-7 细胞，IC50为 250 nM，pIC50为 6.6。
| 生物活性 | Raloxifene 6-Monomethyl Ether (Compound 7) is a Raloxifene derivative that inhibitsestrogen receptorα. Raloxifene 4-Monomethyl Ether inhibits MCF-7 cells with anIC50of 250 nM and apIC50of 6.6[1]. |
体外研究
(In Vitro) | Raloxifene 6-Monomethyl Ether (Compound 7) is a Raloxifene derivative with a methoxy group on C6. Raloxifene 6-Monomethyl Ether holds poor ICsub>50value because of disruption to the hydrogen bond network and steric disfavor[1].
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
