Tiapride 是一种非典型的精神安定剂，是一种选择性多巴胺D2受体拮抗剂，几乎不会引起僵直症状。Tiapride 对 D1，D2，D3，D4 的 IC50值分别为 1440、45.8、>100 和 11.7 μM。
| 生物活性 | Tiapride, an atypical neuroleptic agent, is a selectivedopamine D2-receptorantagonist with little propensity for causing catalepsy and sedation. The IC50values of Tiapride are 1440, 45.8, >100, and 11.7 μM for D1; D2; D3; D4, respectively[1]. |
| IC50& Target | D2Receptor 110-320 nM (IC50) | D3Receptor 180 nM (IC50) |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
