(R)-Verapamil D7 hydrochloride ((R)-(+)-Verapamil D7 hydrochloride) 是 (R)-Verapamil hydrochloride 的一种氘代化合物。(R)-Verapamil hydrochloride ((R)-(+)-Verapamil hydrochloride) 是一种 P-糖蛋白抑制剂。(R)-Verapamil hydrochloride 抑制 MRP1 介导的转运,导致 MRP1 过表达细胞对抗癌药产生化学敏感性。
生物活性 | (R)-Verapamil D7 hydrochloride ((R)-(+)-Verapamil D7 hydrochloride) is a deuterium labeled (R)-Verapamil hydrochloride. (R)-Verapamil hydrochloride ((R)-(+)-Verapamil hydrochloride) is aP-Glycoproteininhibitor. (R)-Verapamil hydrochloride blocks MRP1 mediated transport, resulting in chemosensitization of MRP1-overexpressing cells to anticancer drugs[1][2]. |
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运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |