FXa-IN-1 是一种FXa抑制剂 (IC50: 3 nM,Ki: 0.7 nM)，具有可观的口服生物利用度和半衰期 (in vivo)。FXa-IN-1 可用于血栓栓塞性疾病的研究。
| 生物活性 | FXa-IN-1 is aFXainhibitor (IC50: 3 nM,Ki: 0.7 nM) with respectable oral bioavailability and half-lifein vivo. FXa-IN-1 can be used for thromboembolic disorders[1]. |
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体内研究
(In Vivo) | FXa-IN-1 (compound 22, rats) exhibits good oral bioavailability (F%: 46.9) and half-life (t1/2: 8.8 h, i.v.)[1].
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
