(S)-MRTX-1719 (example 16-7) 是 MRTX-1719 的 S- 对映体。(S)-MRTX-1719 是一种PRMT5/MTA复合物抑制剂,其IC50为7070 nM。
| 生物活性 | (S)-MRTX-1719 (example 16-7) is the S-enantiomer of MRTX-1719. (S)-MRTX-1719 is aPRMT5/MTAcomplex inhibitor, with anIC50of 7070 nM[1]. |
| IC50& Target | IC50: 7070 nM (PRMT5/MTA complex)[1] |
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | | Powder | -20°C | 3 years | | 4°C | 2 years | | In solvent | -80°C | 6 months | | -20°C | 1 month |
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