Ledipasvir diacetone (GS-5885 diacetone) 是 Ledipasvir 的活性药物成分。Ledipasvir 是hepatitis C virus NS5A的有效抑制剂，能够抑制 GT1a 和 GT1b 复制子活性，EC50值分别为 34 pM 和 4 pM。
| 生物活性 | Ledipasvir diacetone (GS-5885 diacetone) is the active ingredient of Ledipasvir. Ledipasvir is an inhibitor of thehepatitis C virus NS5A, withEC50values of 34 pM against GT1a and 4 pM against GT1b replicon. |
体外研究
(In Vitro) | Ledipasvir diacetone is considered the active ingredient, which is converted to Ledipasvir spray-dried dispersion, an amorphous free base.
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
