T-Type calcium channel inhibitor 2 (compound 6g) 是一种有效的T 型钙通道抑制剂，Cav3.1 (α1G)、Cav3.2 (α1H)、Cav3.3 (α1I) (α1H) 的IC50s 分别为31.0、83.1、69.3 μM。T-Type calcium channel inhibitor 2 对 A549、HCT-116 细胞具有细胞毒性，IC50s 分别为5.0、6.4 μM。
| 生物活性 | T-Type calcium channel inhibitor2 (compound 6g) is a potentT-type calcium channelinhibitor withIC50s of 31.0, 83.1, 69.3 μM for Cav3.1 (α1G), Cav3.2 (α1H), Cav3.3 (α1I) (α1H), respectively.T-Type calcium channel inhibitor2 shows cytotoxicity for A549, HCT-116 cells with IC50s of 5.0, 6.4 μM, respectively[1]. |
| IC50& Target[1] | CaV3.1 31.0 μM (IC50) | Cav3.2 83.1 μM (IC50) | CaV3.3 69.3 μM (IC50) |
|
| 分子量 | |
| Formula | |
| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
