BI-3812 是一种高效的BCL6抑制剂,具有抗肿瘤活性,能够抑制 BCL6 的 BTB 结构域,IC50值 ≤3 nM。
产品描述
BI-3812 is an inhibitor of BCL6. Which inhibiting the BTB domain of BCL6 (IC50: 3 nM). BI-3812 also has antitumor activity.
体内活性
BI-3812 is a BCL6 inhibitor, with an IC50 of ≤3 nM. BI-3812 shows an IC50 of 40 nM for the cellular BCL6[1].
Cas No.
2166387-64-8
分子式
C26H32ClN7O5
分子量
558.03
储存和溶解度
DMSO:19.83 mg/mL(35.54 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years