PSB-12062是选择性P2X4拮抗剂，对人类 P2X4 的IC50值为1.38 μM。
产品描述
PSB-12062 is a potent and selective antagonist of P2X4(IC50 of 1.38 μM for human P2X4).
体外活性
PSB-12062 is ?a selective P2X4 antagonist that was equally potent in all three species (IC(50): 0.928-1.76 μM).?The compounds showed an allosteric mechanism of action.
Cas No.
55476-47-6
分子式
C19H15NO3S
分子量
337.39
别名
N-(p-Methylphenylsulfonyl)phenoxazine
储存和溶解度
DMSO:24 mg/mL (71.13mM),Need ultrasonic
Powder: -20°C for 3 years
In solvent: -80°C for 2 years
