Y-29794 Tosylate 是一种具有口服活性、有效且特异性的非肽脯氨酰内肽酶 (PPCE) 抑制剂。
产品描述
Y-29794 Tosylate is an orally active, effective, and specific non-peptide-prolyl endopeptidase (PPCE) inhibitor.
体外活性
Y-29794 Tosylate could penetrate into brain to exhibit dose-dependent and long-lasting inhibition[2].
体内活性
Y-29794 Tosylate selectively and competitively inhibited rat brain PPCE in a reversible manner[2]. Y-29794 Tosylate was found to potentiate the effect of TRH on the release of ACh in the rat hippocampus[2].
Cas No.
143984-17-2
分子式
C30H42N2O4S3
分子量
590.86
别名
Y29794 tosylate;Y 29794;Y29794;Y-29794
储存和溶解度
(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years
