AKR1C1-IN-1 是高选择性AKR1C1抑制剂(Ki:4 nM)。
产品描述
AKR1C1-IN-1 is a human 20α-hydroxysteroid dehydrogenase (AKR1C1) inhibitor (Ki: 4 nM for AKR1C1).
体外活性
AKR1C1-IN-1 inhibits the metabolism of progesterone that in AKR1C1-overexpressed BAECs (IC50:460 nM).
Cas No.
4906-68-7
分子式
C13H9BrO3
分子量
293.11
储存和溶解度
DMSO:10 mM
Powder: -20°C for 3 years
In solvent: -80°C for 2 years
