Racecadotril 是一种中性内肽酶 (NEP) 抑制剂,具有止泻作用。Racecadotril 及其活性代谢物 Thiorphan 抑制小鼠脑中纯化的NEP活性,Ki分别为 4500 和 6.1 nM。
产品描述
Racecadotril has been investigated for the basic science and treatment of Diarrhea, Acute Diarrhea, and Acute Gastroenteritis.
Cas No.
81110-73-8
分子式
C21H23NO4S
分子量
385.48
别名
消旋卡多曲;Acetorphan
储存和溶解度
H2O:<1 mgml
DMSO:21 mg/mL (54.5 mM)
Ethanol:71 mg/mL (184.2 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years