产品描述
LPA2 antagonist 1 is an LPA2 antagonist (IC50: 17 nM).
体外活性
LPA2 antagonist 1 inhibits HCT-116 colon cancer cell proliferation caused by LPA in a doses dependent manner and it also inhibits the phosphorylation of Erk induced by LPA in a concentration-dependent manner .
Cas No.
1017606-66-4
分子式
C20H23Cl2N5O2S2
分子量
500.47
储存和溶解度
DMF:100 mg/mL (199.82 mM)
DMSO:100 mg/mL (199.82 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years