Seglitide acetate 是一种选择性的sst2生长抑素受体激动剂。

Seglitide acetate is a selective agonist of sst2 somatostatin receptor.

Seglitide acetate inhibits [125I]Tyr11-somatostatin-14 binding to rabbit retinal membranes with IC50 of 0.04nM. MK678 stimulated GTPase activity in a concentration-dependent manner with EC50 values of 70.0 ± 16.5 nM, thus supporting the functional coupling between the sst2 somatostatin receptor and the G-proteins.[2].

99248-33-6

C46H60N8O9

869.02

MK-678

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years