6-Bromopravadoline (WIN 54461) 是CB1受体的拮抗剂。6-Bromopravadoline 作为 [3H]Win 55212-2 的结合抑制剂 (IC50=515 nM),反映了其与大麻素受体结合。
产品描述
6-Bromopravadoline (WIN 54461) is an antagonist of CB1. 6-Bromopravadoline acts as an inhibitor of the binding of [3H]Win 55212-2 (IC 50 =515 nM) reflective of cannabinoid receptor binding [1] [2].
Cas No.
166599-63-9
分子式
C23H25BrN2O3
分子量
457.36
别名
WIN 54461
储存和溶解度
DMSO:18.9mg/mL (41.3mM),ultrasonic and warming and heat to 70°C
Powder: -20°C for 3 years
In solvent: -80°C for 2 years