Elagolix sodium 是人GnRH受体拮抗剂，其IC50=0.25 nM，Ki=3.7 nM。
产品描述
Elagolix sodium is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).
体内活性
Elagolix sodium for the treatment of women with moderate to severe endometriosis-associated pain[1]
Cas No.
832720-36-2
分子式
C32H29F5N3NaO5
分子量
653.582
别名
NBI-56418 sodium;恶拉戈利钠
储存和溶解度
DMSO:50 mg/mL (76.50 mM)
H2O:50 mg/mL (76.50 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years
