GRK2-IN-1 hydrochloride(2055990-90-2 free base)

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本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

包装与价格：

包装	价格(元)
1 mg	询价
2 mg	询价
5 mg	询价
10 mg	询价
25 mg	询价
50 mg	询价
100 mg	询价
200 mg	询价
500 mg	询价
1 mL*10 mM(in DMSO)	询价

GRK2-IN-1 hydrochloride

产品描述

GRKs-IN-1 hydrochloride has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50: 130 nM) and GRK5 (IC50: 7.1 μM).

体外活性

GRKs-IN-1 hydrochloride (Compound 14as) is a derivative 14as of paroxetine, shows a 100-fold improvement in cardiomyocyte contractility assays over paroxetine.

Cas No.

T13714L

分子式

C24H26ClFN4O4

分子量

488.94

别名

GRK2-IN-1 hydrochloride

储存和溶解度

DMSO:250 mg/mL (511.31 mM),Need ultrasonic
Powder: -20°C for 3 years
In solvent: -80°C for 2 years