Etifoxine hydrochloride 是GABAA受体亚基 α1β2γ2 和 α1β3γ2 的阳性变构调节剂,是具有 GABA 能的非苯二氮卓类抗焦虑和抗惊厥药物。
产品描述
Etifoxine is an anxiolytic and anticonvulsant drug. Unlike benzodiazepines, etifoxine appears to produce its anxiolytic effects by binding to β2 and β3 subunits of the GABAA receptor complex, and so is acting at a different target site to benzodiazepines, although the physiological effect that is produced is similar to that of benzodiazepines.
Cas No.
56776-32-0
分子式
C17H18Cl2N2O
分子量
337.24
别名
盐酸艾替伏辛;HOE 36-801 hydrochloride
储存和溶解度
DMSO:50 mg/mL (148.26 mM),Need ultrasonic
Powder: -20°C for 3 years
In solvent: -80°C for 2 years