PSB 1115 是一种 A2B 受体拮抗剂，可以抵消 NECA 的抑制作用。
产品描述
PSB 1115 is an A2B receptor antagonist and can counteract the inhibitory effect of NECA.
体外活性
PSB 1115 reversed the decrease in plasma insulin induced by NECA[1].
体内活性
The effect of PSB 1115 was obvious in diabetic GotoKakizaki rats: plasma insulin was increased whereas blood glucose was unchanged. The adenosine levels were not different in normal Wistar rats and in diabetic GotoKakzaki rats[1].
Cas No.
152529-79-8
分子式
C14H14N4O5S
分子量
350.35
储存和溶解度
H2O:<7.77mg/ml
DMSO:<38.84mg/mL
Powder: -20°C for 3 years
In solvent: -80°C for 2 years
