产品描述
PROTAC BRD4 Degrader-1 is an efficacious degrader of BRD4(BRD4 BD1,IC50 of 41.8 nM).
体外活性
PROTAC BRD4 Degrader-1 shows high inhibitory activity against the growth of human monocyte lymphoma cell line THP-1(IC50 value of 0.81 μM), and moderate activity against Raji and HL-60 cell lines[1]
Cas No.
2133360-00-4
分子式
C40H37N9O8
分子量
771.78
储存和溶解度
(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years
