TRPM4-IN-1 是一种有效的阳离子通道TRPM4选择性抑制剂，IC50为 1.5 μM。TRPM4-IN-1 在心脏病和前列腺癌中具有研究价值。

TRPM4-IN-1 is a potent and selective inhibitor of TRPM4 with an IC50 of 1.5 μM.

TRPM4-IN-1 selectively inhibits TRPM4 overexpressed in HEK293 cells. TRPM4-IN-1 inhibits endogenous TRPM4 currents in LNCaP cells. TRPM4-IN-1 restores functional expression of A432T, a loss‐of‐expression TRPM4 variant.

351424-20-9

C15H11Cl2NO4

340.16

CBA;4-chloro-2-(2-(2-chlorophenoxy)acetamido)benzoic acid

DMSO:80mg/ml(235.18mM),Need ultrasonic
Powder: -20°C for 3 years
In solvent: -80°C for 2 years