Tasosartan 是长效血管紧张素 II 受体拮抗剂。
产品描述
Tasosartan is an antagonist of angiotensin II type 2 (AT2) receptor (IC50 = 1.2 nM).
体内活性
In vivo, tasosartan (p.o. or i.v.) blocked by 80% AT1 receptors 1 to 2 h after drug administration and still had a 40% effect at 32 h.
Cas No.
145733-36-4
分子式
C23H21N7O
分子量
411.469
别名
WAY-ANA 756;他索沙坦
储存和溶解度
DMSO:125 mg/mL (303.80 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years
