1-Ethynylpyrene 是有效的细胞色素P450 1A1, 1A2和2B1抑制剂，抑制的IC50分别为 0.18，0.32 和 0.04 μM。
产品描述
1-Ethynylpyrene is an aryl acetylenic inhibitor of CYTP450 1A1(IC50=0.18 μM), 1A2(IC50 = 0.32 μM), and 2B1(IC50 = 0.04 μM).
体外活性
The Ki values of 1-Ethynylpyrene against P450 1A2, and 2B1 is 0.32 and 0.04 μM, respectively[1].
Cas No.
34993-56-1
分子式
C18H10
分子量
226.278
储存和溶解度
DMSO:9.09 mg/mL (40.17 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years
