HA155 是一种高效的 ATX 选择性抑制剂，其IC50=5.7 nM。
产品描述
HA155 selectively and potently inhibits autotaxin with an IC50 of 5.7 nM.
体外活性
HA155 completely attenuates the thrombin-mediated increase in platelet-derived LPA dose-dependently [2].HA155 is an ATX inhibitor by binding to the ATX active site [3].
Cas No.
1312201-00-5
分子式
C24H19BFNO5S
分子量
463.29
别名
CS-963
储存和溶解度
DMSO:8 mg/mL (17.27 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years
