CDK2-IN-4 是选择性的CDK2抑制剂，对 CDK2/cyclin A 的IC50值为 44 nM，选择性高出 CDK1/cyclin B 的 2,000 倍 (IC50=86 μM)。
产品描述
CDK2-IN-4 is a potent and selective inhibitor of CDK2 with an IC50 of 44 nM for CDK2/cyclin A. It shows 2,000-fold selectivity over CDK1/cyclin B with IC50 of 86 uM.
Cas No.
2079895-42-2
分子式
C23H18N6O2S
分子量
442.49
储存和溶解度
DMSO:19.83 mg/mL(44.81 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years
