Cerlapirdine 是一种选择性 5-羟色胺 6 (5-HT6) 受体的完全拮抗剂，用于治疗与阿尔茨海默病和精神分裂症相关的认知障碍。
产品描述
Cerlapirdine is a selective, potent, full antagonist of the 5-hydroxytryptamine 6 (5-HT6) receptor. Cerlapirdine is already in clinical development for the treatment of cognitive disorders related to Alzheimer's disease and schizophrenia. It works by acting as a selective 5-HT6 receptor antagonist.
Cas No.
925448-93-7
分子式
C22H23N3O3S
分子量
409.5
别名
PF05212365;SAM 531;SAM531;PF-05212365;SAM-531;P -05212365;WAY-262,531;Cerlapirdine
储存和溶解度
DMSO:38 mg/mL (92.80 mM),Need ultrasonic and warming and adjust pH to 3 with HCl and heat to 60°C
Powder: -20°C for 3 years
In solvent: -80°C for 2 years
