产品描述
A high affinity blocker for inward-rectifier K+ channels, this compound is a stable derivative of the bee venom toxin tertiapin. Binds to ROMK1 (Kir1.1) and GIRK1/4 (Kir3.1/3.4) channels with high affinity (Ki values are 1.3 and 13.3 nM respectively) and is selective over Kir2.1 channels. Derivative tertiapin LQ also available.
Cas No.
910044-56-3
分子式
C106H175N35O24S4
分子量
2452
别名
Tertiapin-Q
储存和溶解度
H2O:2 mg/mL
Powder: -20°C for 3 years
In solvent: -80°C for 2 years
