GSK2798745 (GSK-2798745) is a novel, first-in-class and potent blocker of transient receptor potential vanilloid 4 (TRPV4) ion channel with the potential to be used for the treatment of pulmonary edema associated with congestive heart failure. It inhibits TRPV4 with IC50s of 1.8 and 1.6 nM for hTRPV4 and rTRPV4, respectively.

纯度：≥98%

CAS：1419609-94-1