生物活性
Bromocriptin mesylate是一种有效的多巴胺受体激动剂，它以最高的亲和力（Ki = 2.5 nM）与D2受体结合。
化学数据
| 目录号 | A13705 |
| 作用机制 | Agonist (激动剂) |
| M. Wt | 750.7 |
| Formula | C32H40BrN5O5CH3SO3H |
| Purity | >99% |
| Storage | Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for36 months.
In solution, store at -20ºC and use within3 monthsto prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles. |
| CAS No. | 22260-51-1 |
| Synonyms | CB 154, Parlodel, Cycloset |
| SMILES | CC(C)C[C@H]1C(=O)N2CCC[C@H]2[C@]3(N1C(=O)[C@](O3)(C(C)C)NC(=O)[C@H]4CN([C@@H]5CC6=C(NC7=CC=CC(=C67)C5=C4)Br)C)O.CS(=O)(=O)O |
储备液配制
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
| 0.1 mM | 13.32 mL | 66.6 mL | 133.21 mL |
| 0.5 mM | 2.66 mL | 13.32 mL | 26.64 mL |
| 1 mM | 1.33 mL | 6.66 mL | 13.32 mL |
| 5 mM | 0.27 mL | 1.33 mL | 2.66 mL |
*The above data is based on the productmolecular weight 750.7. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
