Description: Enalaprilat (also known as MK-422 Dihydrate), the active metabolite of enalapril, is an angiotensin-converting enzyme (ACE) inhibitor with IC50 of 1.94 nM. Enalaprilat has high affinity for human endothelial ACE with IC50 of 1.94 nM and shows bradykinin/angiotensin I selectivity ratio of 1.00 calculated from double displacement experiments.
References: Eur J Pharmacol. 2007 Dec 22;577(1-3):1-6; Br J Anaesth. 2006 Apr;96(4):437-43.
Related CAS#: 76095-16-4 (Enalapril Maleate); 75847-73-3 (Enalapril free base); 149404-21-7 (Enalapril sodium); 349554-02-5 (Enalapril D5 maleate); 349554-00-3 (Enalaprilat D5); 1356922-29-6 (Enalaprilat D5 Sodium)
纯度:≥98%
CAS:76420-72-9