SKF-82958 ((±)-SKF 82958) hydrobromide是多巴胺D1的受体激动剂 (K
0.5=4 nM)，SKF-82958对 D1 受体有选择性(K
0.5=73 nM)。SKF-82958 hydrobromide 诱导大鼠纹状体膜多巴胺 D1 受体依赖性腺苷酸环化酶活性(EC
50=491 nM)。
| 中文别名 | SKF 82958 Hydrobromide;SKF82958 Hydrobromide;74115-01-8 |
| 英文别名 | 3-Allyl-6-chloro-1-phenyl-2,3,4,5-tetrahydro-1H-3-benzazepine-7,8-diol hydrobromide (1:1) |
| CAS号 | 74115-01-8 |
| SMILES | C=CCN1CCC2=C(C(=C(C=C2C(C1)C3=CC=CC=C3)O)O)Cl.Br |
| Inchi | InChI=1S/C19H20ClNO2.BrH/c1-2-9-21-10-8-14-15(11-17(22)19(23)18(14)20)16(12-21)13-6-4-3-5-7-13;/h2-7,11,16,22-23H,1,8-10,12H2;1H |
| InchiKey | WLXGFAVTAAQOFH-UHFFFAOYSA-N |
| 分子式 Formula | C19H20ClNO2 ?HBr |
| 分子量 Molecular Weight | 330 |
| 储藏条件 Storage conditions | storage at -4℃ (1-2weeks), longer storage period at -20℃ (1-2years) |
