WAY 207024 dihydrochloride is a gonadotropin releasing hormone receptor (GnRH-R) antagonist. WAY 207024 dihydrochloride exhibits potent affinity (IC50 are 12 and 71 nM for human and rat GnRH receptors respectively). References: Pelletier JC, Chengalvala MV, Cottom JE, Feingold IB, Green DM, Hauze DB, Huselton CA, Jetter JW, Kopf GS, Lundquist JT, Magolda RL, Mann CW, Mehlmann JF, Rogers JF, Shanno LK, Adams WR, Tio CO, Wrobel JE. Discovery of 6-({4-[2-(4-tert-butylphenyl)-1H-benzimidazol-4-yl]piperazin-1-yl}methyl)quinoxal ine (WAY-207024): an orally active antagonist of the gonadotropin releasing hormone receptor (GnRH-R). J Med Chem. 2009 Apr 9;52(7):2148-52. doi: 10.1021/jm801572m. PubMed PMID: 19271735.

纯度：≥98%

CAS：872002-73-8