NNC-711 is a potent and selective inhibitor of GABA uptake by GAT-1 (IC50 are 0.04, 171, 1700 and 622 μM for hGAT-1, rGAT-2, hGAT-3 and hBGT-1 respectively). NNC-711 is anticonvulsant following systemic administration in vivo. References: Viereckel T, Kostic M, Bahner F, Draguhn A, Both M. Effects of the GABA-uptake blocker NNC-711 on spontaneous sharp wave-ripple complexes in mouse hippocampal slices. Hippocampus. 2013 May;23(5):323-9. doi: 10.1002/hipo.22104. Epub 2013 Mar 5. PubMed PMID: 23460368.

纯度：≥98%

CAS：159094-94-7